Product

THIS PRODUCT IS FOR RESEARCH PURPOSES ONLY.

+ Description

PT-141 is the isomer of Melanotan 2 without the C-end amide group, which avoids characteristics such as sunburn stimulation and enhances characteristics such as libido stimulation. Bremelanotide belongs to the category of melanocortinagonists. PT-141 does not affect the vascular system and its selective effect is limited to activation and stimulation of melanocortin receptors to increase libido and and sexual appeal.

PT-141 is a sterile, non-pyrogenic, white lyophilized powder intended for subcutaneous or intramuscular injection, after reconstitution with sterile Water for Injection (0,3% m-Cresol).

Molecular Weight: 9111.6 daltons – confirmed by Mass Spectrometry. It is produced in E. coli using a patented expression system the IGF-I Long[R3] is correctly folded and purified by several chromatography steps to yield Receptor Grade IGF-I Long[R3].

IGF-1 L[R3] is a sterile, non-pyrogenic, white lyophilized powder intended for subcutaneous or intramuscular injection, after reconstitution with sterile Water for injection ( 0.3% m-Cresol).

+ Mechanism of action

PT-141 is considered as a synthetic aphrodisiac. Alternatively to Viagra and Cialis, it has no influence upon the vascular system, but directly increases sexual desire.

PT-141 activates the melanocortin receptors MC1R and MC4R in the central nervous system, modulates inflammation and reduces the restriction in blood supply to the tissues. PT-141 is a deaminated derivative and metabolite of Melanotan II. PT-141 also acts as an agonist. PT-141 has proved its safeness and efficiency on a broad range of patients.

+ Adverse reaction

PT-141 (Bremelanotide) is considered to be much safer compared to Viagra or Cialis. However, as all other medicine it might be the reason of several adverse reactions to occur, such as nausea, decreased appetite; flushing of the face and increased blood pressure.

The last one should not cause discomfort for healthy individuals. Injectable PT-141 is considered not to have this particular minor effect.

+ Instructions for reconstitution

The injection is given into the sub-cutaneous layer which includes adipose tissue (fat).

If you are using insulin syringes which have short needles, you will need to enter the skin at 90°. to the skin, otherwise you can inject as shown in the illustration above with a 29 or 30 gauge, 0.5" needle.

+ Dosage

Recommended dosage of PT-141: 0.30 mg (trial) – 0.70 mg (average) – 1 mg (optimal) – 1.5 mg (strong), 45 – 60 mins before sex.

+ Storage

• This product can be used not more than 3 years from the production date (see box).
• After reconstitution, may be stored for a maximum of 14 days in a refrigirator at 2°C – 8°C.
• Store vials in an upright position.
• Store in a refrigerator (2°C – 8°C). Keep in the outer carton in order to protect from light.
• For one month can be stored at room temperature.